Preparation and Cyclodextrin Solubilization of the Antibacterial Agent Benzoyl Metronidazole
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چکیده
منابع مشابه
Preparation and Cyclodextrin Solubilization of the Antibacterial Agent Benzoyl Metronidazole
A one-pot method for the preparation of benzoyl metronidazole was achieved by using N,N'-carbonyldiimidazole as a coupling reagent. Moreover, it was found that the byproduct imidazole as the catalyst promoted the reaction. In addition, the β-cyclodextrin solubilization of benzoyl metronidazole was investigated by phase-solubility method. The phase-solubility studies indicated that the solubilit...
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Evaluation of cyclodextrin solubilization of drugs.
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ژورنال
عنوان ژورنال: The Scientific World Journal
سال: 2013
ISSN: 1537-744X
DOI: 10.1155/2013/306476